???pagination.result.count???
Agonist pharmacology of two Drosophila GABA receptor splice variants. , Hosie AM, Sattelle DB., Br J Pharmacol. December 1, 1996; 119 (8): 1577-85.
Actions of picrodendrin antagonists on dieldrin-sensitive and -resistant Drosophila GABA receptors. , Hosie AM, Ozoe Y, Koike K, Ohmoto T, Nikaido T, Sattelle DB., Br J Pharmacol. December 1, 1996; 119 (8): 1569-76.
Allosteric modulation by single enantiomers of a C3-chiral 1,4-benzodiazepine of the gamma aminobutyric acid type A receptor channel expressed in Xenopus oocytes. , Demuro A, Burgio M, Berton F, Francesconi W, Bertucci C., Chirality. January 1, 1997; 9 (3): 286-90.
Neuroendocrine gamma-aminobutyric acid (GABA): functional differences in GABAA versus GABAB receptor inhibition of the melanotrope cell of Xenopus laevis. , Buzzi M, Bemelmans FF, Roubos EW , Jenks BG ., Endocrinology. January 1, 1997; 138 (1): 203-12.
Neuroendocrine γ-Aminobutyric Acid (GABA): Functional Differences in GABAA Versus GABAB Receptor Inhibition of the Melanotrope Cell of Xenopus laevis1. , Buzzi M, Bemelmans FF, Roubos EW , Jenks BG ., Endocrinology. January 1, 1997; 138 (1): 203-212.
3 alpha-Hydroxy-3 beta-(phenylethynyl)-5 beta-pregnan-20-ones: synthesis and pharmacological activity of neuroactive steroids with high affinity for GABAA receptors. , Upasani RB, Yang KC, Acosta-Burruel M, Konkoy CS, McLellan JA, Woodward RM, Lan NC, Carter RB, Hawkinson JE., J Med Chem. January 3, 1997; 40 (1): 73-84.
Synthesis and in vitro activity of 3 beta-substituted-3 alpha-hydroxypregnan-20-ones: allosteric modulators of the GABAA receptor. , Hogenkamp DJ, Tahir SH, Hawkinson JE, Upasani RB, Alauddin M, Kimbrough CL, Acosta-Burruel M, Whittemore ER, Woodward RM, Lan NC, Gee KW, Bolger MB., J Med Chem. January 3, 1997; 40 (1): 61-72.
Both GABAA and GABAB receptors participate in suppression of [CA2+]i pulsing in toad melanotrophs. , Shibuya I, Kongsamut S, Douglas WW., Eur J Pharmacol. February 26, 1997; 321 (2): 241-6.
Subunit-dependent interaction of the general anaesthetic etomidate with the gamma-aminobutyric acid type A receptor. , Hill-Venning C, Belelli D, Peters JA, Lambert JJ., Br J Pharmacol. March 1, 1997; 120 (5): 749-56.
Differential sensitivities of mammalian neuronal and muscle nicotinic acetylcholine receptors to general anesthetics. , Violet JM, Downie DL, Nakisa RC, Lieb WR, Franks NP., Anesthesiology. April 1, 1997; 86 (4): 866-74.
Alpha 4 beta 2 neuronal nicotinic acetylcholine receptors in the central nervous system are inhibited by isoflurane and propofol, but alpha 7-type nicotinic acetylcholine receptors are unaffected. , Flood P, Ramirez-Latorre J, Role L., Anesthesiology. April 1, 1997; 86 (4): 859-65.
Ethanol, flunitrazepam, and pentobarbital modulation of GABAA receptors expressed in mammalian cells and Xenopus oocytes. , Harris RA, Mihic SJ, Brozowski S, Hadingham K, Whiting PJ., Alcohol Clin Exp Res. May 1, 1997; 21 (3): 444-51.
Subtle changes in residue 77 of the gamma subunit of alpha1beta2gamma2 GABAA receptors drastically alter the affinity for ligands of the benzodiazepine binding site. , Buhr A, Baur R, Sigel E., J Biol Chem. May 2, 1997; 272 (18): 11799-804.
Neuronally restricted RNA splicing regulates the expression of a novel GABAA receptor subunit conferring atypical functional properties [corrected; erratum to be published]. , Whiting PJ, McAllister G, Vassilatis D, Bonnert TP, Heavens RP, Smith DW, Hewson L, O'Donnell R, Rigby MR, Sirinathsinghji DJ, Marshall G, Thompson SA, Wafford KA, Vasilatis D., J Neurosci. July 1, 1997; 17 (13): 5027-37.
Synaptic transmission in the pineal eye of young Xenopus laevis tadpoles: a role for NMDA and non-NMDA glutamate and non-glutaminergic receptors? , Jamieson D., J Comp Physiol A. August 1, 1997; 181 (2): 177-86.
A point mutation in the gamma2 subunit of gamma-aminobutyric acid type A receptors results in altered benzodiazepine binding site specificity. , Buhr A, Sigel E., Proc Natl Acad Sci U S A. August 5, 1997; 94 (16): 8824-9.
Inhibitory effects of corymine, an alkaloidal component from the leaves of Hunteria zeylanica, on glycine receptors expressed in Xenopus oocytes. , Leewanich P, Tohda M, Matsumoto K , Subhadhirasakul S, Takayama H, Aimi N, Watanabe H., Eur J Pharmacol. August 13, 1997; 332 (3): 321-6.
Synthesis and binding affinity of 2-phenylimidazo[1,2-alpha]pyridine derivatives for both central and peripheral benzodiazepine receptors. A new series of high-affinity and selective ligands for the peripheral type. , Trapani G, Franco M, Ricciardi L, Latrofa A, Genchi G, Sanna E, Tuveri F, Cagetti E, Biggio G, Liso G., J Med Chem. September 12, 1997; 40 (19): 3109-18.
The interaction of the general anesthetic etomidate with the gamma-aminobutyric acid type A receptor is influenced by a single amino acid. , Belelli D, Lambert JJ, Peters JA, Wafford K, Whiting PJ., Proc Natl Acad Sci U S A. September 30, 1997; 94 (20): 11031-6.
Residues at positions 206 and 209 of the alpha1 subunit of gamma-aminobutyric AcidA receptors influence affinities for benzodiazepine binding site ligands. , Buhr A, Schaerer MT, Baur R, Sigel E., Mol Pharmacol. October 1, 1997; 52 (4): 676-82.
Pre- and postsynaptic modulation of spinal GABAergic neurotransmission by the neurosteroid, 5 beta-pregnan-3 alpha-ol-20-one. , Reith CA, Sillar KT ., Dev Biol. October 3, 1997; 770 (1-2): 202-12.
Key amino acids in the gamma subunit of the gamma-aminobutyric acidA receptor that determine ligand binding and modulation at the benzodiazepine site. , Wingrove PB, Thompson SA, Wafford KA, Whiting PJ., Mol Pharmacol. November 1, 1997; 52 (5): 874-81.
The interaction of general anaesthetics with recombinant GABAA and glycine receptors expressed in Xenopus laevis oocytes: a comparative study. , Pistis M, Belelli D, Peters JA, Lambert JJ., Br J Pharmacol. December 1, 1997; 122 (8): 1707-19.
Analogues of gamma-aminobutyric acid (GABA) and trans-4-aminocrotonic acid (TACA) substituted in the 2 position as GABAC receptor antagonists. , Chebib M, Vandenberg RJ, Johnston GA ., Br J Pharmacol. December 1, 1997; 122 (8): 1551-60.
Differences in agonist/antagonist binding affinity and receptor transduction using recombinant human gamma-aminobutyric acid type A receptors. , Ebert B, Thompson SA, Saounatsou K, McKernan R, Krogsgaard-Larsen P, Wafford KA., Mol Pharmacol. December 1, 1997; 52 (6): 1150-6.
Identification of a Zn2+ binding site on the murine GABAA receptor complex: dependence on the second transmembrane domain of beta subunits. , Wooltorton JR, McDonald BJ, Moss SJ, Smart TG., J Physiol. December 15, 1997; 505 ( Pt 3) 633-40.
Characterization of the hyperpolarization-activated chloride current in dissociated rat sympathetic neurons. , Clark S, Jordt SE, Jentsch TJ, Mathie A., J Physiol. February 1, 1998; 506 ( Pt 3) 665-78.
Modulatory and direct effects of propofol on recombinant GABAA receptors expressed in xenopus oocytes: influence of alpha- and gamma2-subunits. , Lam DW, Reynolds JN., Dev Biol. February 16, 1998; 784 (1-2): 179-87.
Characterization and comparative pharmacological studies of a functional gamma-aminobutyric acid (GABA) receptor cloned from the tobacco budworm, Heliothis virescens (Noctuidae:Lepidoptera). , Wolff MA, Wingate VP., Invert Neurosci. March 1, 1998; 3 (4): 305-15.
Interaction of H+ and Zn2+ on recombinant and native rat neuronal GABAA receptors. , Krishek BJ, Moss SJ, Smart TG., J Physiol. March 15, 1998; 507 ( Pt 3) (Pt 3): 639-52.
Cloning and functional expression of alternative spliced variants of the rho1 gamma-aminobutyrate receptor. , Martínez-Torres A, Vazquez AE, Panicker MM, Miledi R ., Proc Natl Acad Sci U S A. March 31, 1998; 95 (7): 4019-22.
Gamma subunit dependent modulation by nitric oxide (NO) in recombinant GABAA receptor. , Fukami S, Uchida I, Mashimo T, Takenoshita M, Yoshiya I., Neuroreport. April 20, 1998; 9 (6): 1089-92.
Molecular composition of GABAC receptors. , Enz R, Cutting GR., Vision Res. May 1, 1998; 38 (10): 1431-41.
Enhancement of gamma-aminobutyric acidA receptor activity by alpha-chloralose. , Garrett KM, Gan J., J Pharmacol Exp Ther. May 1, 1998; 285 (2): 680-6.
Propofol analogues. Synthesis, relationships between structure and affinity at GABAA receptor in rat brain, and differential electrophysiological profile at recombinant human GABAA receptors. , Trapani G, Latrofa A, Franco M, Altomare C, Sanna E, Usala M, Biggio G, Liso G., J Med Chem. May 21, 1998; 41 (11): 1846-54.
GABAA-benzodiazepine receptors in the striatum are involved in the sedation produced by a moderate, but not an intoxicating ethanol dose in outbred Wistar rats. , June HL, Cason CR, Cheatham G, Lui R, Gan T, Cook JM., Dev Biol. May 25, 1998; 794 (1): 103-18.
[Zinc modulation of GABA receptors expressed in Xenopus oocytes injected with carp brain poly(A)+ RNA]. , Bai XC, Bao YD., Sheng Li Xue Bao. June 1, 1998; 50 (3): 268-74.
Functional characterization and visualization of a GABAA receptor-GFP chimera expressed in Xenopus oocytes. , Bueno OF, Robinson LC, Alvarez-Hernandez X, Leidenheimer NJ., Brain Res Mol Brain Res. August 31, 1998; 59 (2): 165-77.
Substituted 3beta-phenylethynyl derivatives of 3alpha-hydroxy-5alpha-pregnan-20-one: remarkably potent neuroactive steroid modulators of gamma-aminobutyric acidA receptors. , Hawkinson JE, Acosta-Burruel M, Yang KC, Hogenkamp DJ, Chen JS , Lan NC, Drewe JA, Whittemore ER, Woodward RM, Carter RB, Upasani RB., J Pharmacol Exp Ther. October 1, 1998; 287 (1): 198-207.
A GABAA receptor alpha1 subunit tagged with green fluorescent protein requires a beta subunit for functional surface expression. , Connor JX, Boileau AJ, Czajkowski C., J Biol Chem. October 30, 1998; 273 (44): 28906-11.
Inhibition of GABAA receptor function by tyrosine kinase inhibitors and their inactive analogues. , Dunne EL, Moss SJ, Smart TG., Mol Cell Neurosci. November 1, 1998; 12 (4-5): 300-10.
Activation of protein kinase C induces gamma-aminobutyric acid type A receptor internalization in Xenopus oocytes. , Chapell R, Bueno OF, Alvarez-Hernandez X, Robinson LC, Leidenheimer NJ., J Biol Chem. December 4, 1998; 273 (49): 32595-601.
Molecular and neurochemical evaluation of the effects of etizolam on GABAA receptors under normal and stress conditions. , Sanna E, Pau D, Tuveri F, Massa F, Maciocco E, Acquas C, Floris C, Fontana SN, Maira G, Biggio G., Arzneimittelforschung. February 1, 1999; 49 (2): 88-95.
Complementary regulation of anaesthetic activation of human (alpha6beta3gamma2L) and Drosophila (RDL) GABA receptors by a single amino acid residue. , Pistis M, Belelli D, McGurk K, Peters JA, Lambert JJ., J Physiol. February 15, 1999; 515 ( Pt 1) 3-18.
Subunit dependent modulation of GABAA receptor function by neuroactive steroids. , Maitra R, Reynolds JN., Dev Biol. February 20, 1999; 819 (1-2): 75-82.
Potentiation of GABAA receptors expressed in Xenopus oocytes by perfume and phytoncid. , Aoshima H, Hamamoto K., Biosci Biotechnol Biochem. April 1, 1999; 63 (4): 743-8.
In vivo and in vitro toxicodynamic analyses of new quinolone-and nonsteroidal anti-inflammatory drug-induced effects on the central nervous system. , Kita H, Matsuo H, Takanaga H, Kawakami J, Yamamoto K, Iga T, Naito M, Tsuruo T, Asanuma A, Yanagisawa K, Sawada Y., Antimicrob Agents Chemother. May 1, 1999; 43 (5): 1091-7.
Sulfated and unsulfated steroids modulate gamma-aminobutyric acidA receptor function through distinct sites. , Park-Chung M, Malayev A, Purdy RH, Gibbs TT, Farb DH., Dev Biol. May 29, 1999; 830 (1): 72-87.
A single amino acid confers barbiturate sensitivity upon the GABA rho 1 receptor. , Belelli D, Pau D, Cabras G, Peters JA, Lambert JJ., Br J Pharmacol. June 1, 1999; 127 (3): 601-4.
Residues in transmembrane domains I and II determine gamma-aminobutyric acid type AA receptor subtype-selective antagonism by furosemide. , Thompson SA, Arden SA, Marshall G, Wingrove PB, Whiting PJ, Wafford KA., Mol Pharmacol. June 1, 1999; 55 (6): 993-9.