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Characterization of a novel α-conotoxin from conus textile that selectively targets α6/α3β2β3 nicotinic acetylcholine receptors. , Luo S., J Biol Chem. January 11, 2013; 288 (2): 894-902.
Fast silencing reveals a lost role for reciprocal inhibition in locomotion. , Moult PR., Neuron. January 9, 2013; 77 (1): 129-40.
Toxicity of the synthetic polymeric 3-alkylpyridinium salt (APS3) is due to specific block of nicotinic acetylcholine receptors. , Grandič M., Toxicology. January 7, 2013; 303 25-33.
Blocking of the human ether-à- go-go-related gene channel by imatinib mesylate. , Dong Q., Biol Pharm Bull. January 1, 2013; 36 (2): 268-75.
The neuroplastin adhesion molecules are accessory proteins that chaperone the monocarboxylate transporter MCT2 to the neuronal cell surface. , Wilson MC., PLoS One. January 1, 2013; 8 (11): e78654.
A natural point mutation changes both target selectivity and mechanism of action of sea anemone toxins. , Peigneur S., FASEB J. December 1, 2012; 26 (12): 5141-51.
Inhibitory effect of the recombinant Phoneutria nigriventer Tx1 toxin on voltage-gated sodium channels. , Silva AO ., Biochimie. December 1, 2012; 94 (12): 2756-63.
The non-competitive acetylcholinesterase inhibitor APS12-2 is a potent antagonist of skeletal muscle nicotinic acetylcholine receptors. , Grandič M., Toxicol Appl Pharmacol. December 1, 2012; 265 (2): 221-8.
Mixed antagonistic effects of the ginkgolides at recombinant human ρ1 GABAC receptors. , Huang SH., Neuropharmacology. November 1, 2012; 63 (6): 1127-39.
Novel electrophysiological properties of dronedarone: inhibition of human cardiac two-pore-domain potassium (K2P) channels. , Schmidt C., Naunyn Schmiedebergs Arch Pharmacol. October 1, 2012; 385 (10): 1003-16.
Cartilage on the move: cartilage lineage tracing during tadpole metamorphosis. , Kerney RR., Dev Growth Differ. October 1, 2012; 54 (8): 739-52.
Differentiating enantioselective actions of GABOB: a possible role for threonine 244 in the binding site of GABA(C) ρ(1) receptors. , Yamamoto I., ACS Chem Neurosci. September 19, 2012; 3 (9): 665-73.
Design of bioactive peptides from naturally occurring μ-conotoxin structures. , Stevens M., J Biol Chem. September 7, 2012; 287 (37): 31382-92.
N3,N7-diaminophenothiazinium derivatives as antagonists of α7-nicotinic acetylcholine receptors expressed in Xenopus oocytes. , Sadek B., Pharmacol Res. September 1, 2012; 66 (3): 213-8.
Active intestinal absorption of fluoroquinolone antibacterial agent ciprofloxacin by organic anion transporting polypeptide, Oatp1a5. , Arakawa H., Biopharm Drug Dispos. September 1, 2012; 33 (6): 332-41.
Tuning of EAG K(+) channel inactivation: molecular determinants of amplification by mutations and a small molecule. , Garg V., J Gen Physiol. September 1, 2012; 140 (3): 307-24.
Azemiopsin from Azemiops feae viper venom, a novel polypeptide ligand of nicotinic acetylcholine receptor. , Utkin YN., J Biol Chem. August 3, 2012; 287 (32): 27079-86.
Inhibition of cardiac Kir2.1-2.3 channels by beta3 adrenoreceptor antagonist SR 59230A. , Kulzer M., Biochem Biophys Res Commun. July 27, 2012; 424 (2): 315-20.
Inhibitory effects of dextrorotatory morphinans on the human 5-HT(3A) receptor expressed in Xenopus oocytes: Involvement of the N-terminal domain of the 5-HT(3A) receptor. , Lee BH., Eur J Pharmacol. July 5, 2012; 686 (1-3): 41-9.
Open-channel blockade is less effective on GluN3B than GluN3A subunit-containing NMDA receptors. , McClymont DW., Eur J Pharmacol. July 5, 2012; 686 (1-3): 22-31.
Mutation conferring apical-targeting motif on AE1 exchanger causes autosomal dominant distal RTA. , Fry AC., J Am Soc Nephrol. July 1, 2012; 23 (7): 1238-49.
A novel µ-conopeptide, CnIIIC, exerts potent and preferential inhibition of NaV1.2/1.4 channels and blocks neuronal nicotinic acetylcholine receptors. , Favreau P., Br J Pharmacol. July 1, 2012; 166 (5): 1654-68.
Probing the Xenopus laevis inner ear transcriptome for biological function. , Powers TR ., BMC Genomics. June 8, 2012; 13 225.
18β-Glycyrrhetinic acid preferentially blocks late Na current generated by ΔKPQ Nav1.5 channels. , Du YM., Acta Pharmacol Sin. June 1, 2012; 33 (6): 752-60.
Pharmacological characterization of the Haemonchus contortus GABA-gated chloride channel, Hco-UNC-49: modulation by macrocyclic lactone anthelmintics and a receptor for piperazine. , Brown DD ., Vet Parasitol. April 30, 2012; 185 (2-4): 201-9.
TASK1 (K(2P)3.1) K(+) channel inhibition by endothelin-1 is mediated through Rho kinase-dependent phosphorylation. , Seyler C., Br J Pharmacol. March 1, 2012; 165 (5): 1467-75.
Understanding ciliated epithelia: the power of Xenopus. , Werner ME., Genesis. March 1, 2012; 50 (3): 176-85.
Structure-activity relationships for allosteric NMDA receptor inhibitors based on 2-naphthoic acid. , Costa BM., Neuropharmacology. March 1, 2012; 62 (4): 1730-6.
[Mg(2+) inhibits ATP-activated current mediated by rat P2X4 receptors expressed in Xenopus oocytes]. , Peng F., Sheng Li Xue Bao. February 25, 2012; 64 (1): 75-81.
The inhibitory potency of local anesthetics on NMDA receptor signalling depends on their structural features. , Gronwald C., Eur J Pharmacol. January 5, 2012; 674 (1): 13-9.
Molecular basis of selective antagonism of the P2X1 receptor for ATP by NF449 and suramin: contribution of basic amino acids in the cysteine-rich loop. , El-Ajouz S., Br J Pharmacol. January 1, 2012; 165 (2): 390-400.
Role of human nucleoside transporters in the uptake and cytotoxicity of azacitidine and decitabine. , Damaraju VL., Nucleosides Nucleotides Nucleic Acids. January 1, 2012; 31 (3): 236-55.
γ-Aminobutyric acid transporter 2 mediates the hepatic uptake of guanidinoacetate, the creatine biosynthetic precursor, in rats. , Tachikawa M., PLoS One. January 1, 2012; 7 (2): e32557.
Cloning and characterization of a P2X receptor expressed in the central nervous system of Lymnaea stagnalis. , Bavan S., PLoS One. January 1, 2012; 7 (11): e50487.
Chromatin modification by PSC occurs at one PSC per nucleosome and does not require the acidic patch of histone H2A. , Lo SM., PLoS One. January 1, 2012; 7 (10): e47162.
A molecular switch driving inactivation in the cardiac K+ channel HERG. , Köpfer DA., PLoS One. January 1, 2012; 7 (7): e41023.
Complement fragment C3a controls mutual cell attraction during collective cell migration. , Carmona-Fontaine C., Dev Cell. December 13, 2011; 21 (6): 1026-37.
Interaction of bupropion and zinc with neuronal nicotinic acetylcholine receptors. , García-Colunga J., Neuropharmacology. December 1, 2011; 61 (8): 1202-9.
The influence of calcium ions on nickel modulation of NMDA receptor currents. , Gavazzo P., Metallomics. December 1, 2011; 3 (12): 1376-83.
Functional characterization and high-throughput screening of positive allosteric modulators of α7 nicotinic acetylcholine receptors in IMR-32 neuroblastoma cells. , Gopalakrishnan SM., Assay Drug Dev Technol. December 1, 2011; 9 (6): 635-45.
Discovery, characterization, and structure-activity relationships of an inhibitor of inward rectifier potassium (Kir) channels with preference for Kir2.3, Kir3.x, and Kir7.1. , Raphemot R., Front Pharmacol. November 30, 2011; 2 75.
Postsynaptic TRPC1 function contributes to BDNF-induced synaptic potentiation at the developing neuromuscular junction. , McGurk JS., J Neurosci. October 12, 2011; 31 (41): 14754-62.
Varenicline is a potent agonist of the human 5-hydroxytryptamine3 receptor. , Lummis SC., J Pharmacol Exp Ther. October 1, 2011; 339 (1): 125-31.
Molecular determinants for activation of human ether-à- go-go-related gene 1 potassium channels by 3-nitro-n-(4-phenoxyphenyl) benzamide. , Garg V., Mol Pharmacol. October 1, 2011; 80 (4): 630-7.
Split-inteins for simultaneous, site-specific conjugation of quantum dots to multiple protein targets in vivo. , Charalambous A., J Nanobiotechnology. September 15, 2011; 9 37.
Expression of organic anion-transporting polypeptides 1B1 and 1B3 in ovarian cancer cells: relevance for paclitaxel transport. , Svoboda M., Biomed Pharmacother. September 1, 2011; 65 (6): 417-26.
Importance of position 8 in μ-conotoxin KIIIA for voltage-gated sodium channel selectivity. , Van Der Haegen A., FEBS J. September 1, 2011; 278 (18): 3408-18.
Effects of the histamine H(1) receptor antagonist hydroxyzine on hERG K(+) channels and cardiac action potential duration. , Lee BH., Acta Pharmacol Sin. September 1, 2011; 32 (9): 1128-37.
Extracellular potassium inhibits Kv7.1 potassium channels by stabilizing an inactivated state. , Larsen AP., Biophys J. August 17, 2011; 101 (4): 818-27.
External Cu2+ inhibits human epithelial Na+ channels by binding at a subunit interface of extracellular domains. , Chen J ., J Biol Chem. August 5, 2011; 286 (31): 27436-46.