???pagination.result.count???
Inhibitory Effects of Quercetin on Muscle-type of Nicotinic Acetylcholine Receptor-Mediated Ion Currents Expressed in Xenopus Oocytes. , Lee BH., Korean J Physiol Pharmacol. August 1, 2011; 15 (4): 195-201.
Carvedilol targets human K2P 3.1 ( TASK1) K+ leak channels. , Staudacher K., Br J Pharmacol. July 1, 2011; 163 (5): 1099-110.
A bifunctional sea anemone peptide with Kunitz type protease and potassium channel inhibiting properties. , Peigneur S., Biochem Pharmacol. July 1, 2011; 82 (1): 81-90.
Multiple inhibitory actions of lidocaine on Torpedo nicotinic acetylcholine receptors transplanted to Xenopus oocytes. , Alberola-Die A., J Neurochem. June 1, 2011; 117 (6): 1009-19.
Mutations of the same conserved glutamate residue in NBD2 of the sulfonylurea receptor 1 subunit of the KATP channel can result in either hyperinsulinism or neonatal diabetes. , Männikkö R., Diabetes. June 1, 2011; 60 (6): 1813-22.
In vitro risk assessment of AZD9056 perpetrating a transporter-mediated drug-drug interaction with methotrexate. , Elsby R., Eur J Pharm Sci. May 18, 2011; 43 (1-2): 41-9.
Developing potent human uric acid transporter 1 (hURAT1) inhibitors. , Wempe MF., J Med Chem. April 28, 2011; 54 (8): 2701-13.
A constitutive pan-hexose permease for the Plasmodium life cycle and transgenic models for screening of antimalarial sugar analogs. , Blume M., FASEB J. April 1, 2011; 25 (4): 1218-29.
Cloning and characterization of GABAA α subunits and GABAB subunits in Xenopus laevis during development. , Kaeser GE., Dev Dyn. April 1, 2011; 240 (4): 862-73.
Effects of diltiazem and propafenone on the inactivation and recovery kinetics of fKv1.4 channel currents expressed in Xenopus oocytes. , Zhang D., Acta Pharmacol Sin. April 1, 2011; 32 (4): 465-77.
A fungal metabolite asperparaline a strongly and selectively blocks insect nicotinic acetylcholine receptors: the first report on the mode of action. , Hirata K., PLoS One. April 1, 2011; 6 (4): e18354.
The penultimate arginine of the carboxyl terminus determines slow desensitization in a P2X receptor from the cattle tick Boophilus microplus. , Bavan S., Mol Pharmacol. April 1, 2011; 79 (4): 776-85.
Transdifferentiation of tadpole pancreatic acinar cells to duct cells mediated by Notch and stromelysin-3. , Mukhi S ., Dev Biol. March 15, 2011; 351 (2): 311-7.
Embryonic frog epidermis: a model for the study of cell-cell interactions in the development of mucociliary disease. , Dubaissi E ., Dis Model Mech. March 1, 2011; 4 (2): 179-92.
Discovery of potent competitive antagonists and positive modulators of the P2X2 receptor. , Baqi Y., J Med Chem. February 10, 2011; 54 (3): 817-30.
The N-terminal coiled-coil of Ndel1 is a regulated scaffold that recruits LIS1 to dynein. , Zyłkiewicz E., J Cell Biol. February 7, 2011; 192 (3): 433-45.
Directed differentiation of human pluripotent stem cells into intestinal tissue in vitro. , Spence JR., Nature. February 3, 2011; 470 (7332): 105-9.
Raltegravir is a substrate for SLC22A6: a putative mechanism for the interaction between raltegravir and tenofovir. , Moss DM., Antimicrob Agents Chemother. February 1, 2011; 55 (2): 879-87.
Effects of a highly selective acetylcholine-activated K+ channel blocker on experimental atrial fibrillation. , Machida T., Circ Arrhythm Electrophysiol. February 1, 2011; 4 (1): 94-102.
Specification of ion transport cells in the Xenopus larval skin. , Quigley IK ., Development. February 1, 2011; 138 (4): 705-14.
Quercetin Inhibits α3β4 Nicotinic Acetylcholine Receptor-Mediated Ion Currents Expressed in Xenopus Oocytes. , Lee BH., Korean J Physiol Pharmacol. February 1, 2011; 15 (1): 17-22.
Molecular diversity and functional evolution of scorpion potassium channel toxins. , Zhu S., Mol Cell Proteomics. February 1, 2011; 10 (2): M110.002832.
Amino acid derivatives are substrates or non-transported inhibitors of the amino acid transporter PAT2 (slc36a2). , Edwards N ., Biochim Biophys Acta. January 1, 2011; 1808 (1): 260-70.
Ginkgolide B and bilobalide block the pore of the 5-HT₃receptor at a location that overlaps the picrotoxin binding site. , Thompson AJ., Neuropharmacology. January 1, 2011; 60 (2-3): 488-95.
Quantification of the Mg2+-induced potency shift of amantadine and memantine voltage-dependent block in human recombinant GluN1/GluN2A NMDARs. , Otton HJ., Neuropharmacology. January 1, 2011; 60 (2-3): 388-96.
Acquisition of glial cells missing 2 enhancers contributes to a diversity of ionocytes in zebrafish. , Shono T., PLoS One. January 1, 2011; 6 (8): e23746.
A potent potassium channel blocker from Mesobuthus eupeus scorpion venom. , Gao B., Biochimie. December 1, 2010; 92 (12): 1847-53.
α-Conotoxin BuIA[T5A;P6O]: a novel ligand that discriminates between α6ß4 and α6ß2 nicotinic acetylcholine receptors and blocks nicotine-stimulated norepinephrine release. , Azam L., FASEB J. December 1, 2010; 24 (12): 5113-23.
Aminoglycoside block of P2X2 receptors heterologously expressed in Xenopus laevis oocytes. , Bongartz EV., Purinergic Signal. December 1, 2010; 6 (4): 393-403.
Open channel block of the fast transient outward K+ current by primaquine and chloroquine in rat left ventricular cardiomyocytes. , Wagner M., Eur J Pharmacol. November 25, 2010; 647 (1-3): 13-20.
The effect of Δ9-tetrahydrocannabinol on 5-HT3 receptors depends on the current density. , Yang KH., Neuroscience. November 24, 2010; 171 (1): 40-9.
Inhibition of thyroid hormone release from cultured amphibian thyroid glands by methimazole, 6-propylthiouracil, and perchlorate. , Hornung MW., Toxicol Sci. November 1, 2010; 118 (1): 42-51.
Inhibition of TRPV1 for the treatment of sensitive skin. , Kueper T., Exp Dermatol. November 1, 2010; 19 (11): 980-6.
Assessment of structurally diverse philanthotoxin analogues for inhibitory activity on ionotropic glutamate receptor subtypes: discovery of nanomolar, nonselective, and use-dependent antagonists. , Frølund S., J Med Chem. October 28, 2010; 53 (20): 7441-51.
The inhibition of monocarboxylate transporter 2 ( MCT2) by AR-C155858 is modulated by the associated ancillary protein. , Ovens MJ., Biochem J. October 15, 2010; 431 (2): 217-25.
Identification of selective norbornane-type aspartate analogue inhibitors of the glutamate transporter 1 ( GLT-1) from the chemical universe generated database (GDB). , Luethi E., J Med Chem. October 14, 2010; 53 (19): 7236-50.
Development of a novel selective inhibitor of the Down syndrome-related kinase Dyrk1A. , Ogawa Y., Nat Commun. October 5, 2010; 1 86.
Intestinal absorption of HMG-CoA reductase inhibitor pravastatin mediated by organic anion transporting polypeptide. , Shirasaka Y., Pharm Res. October 1, 2010; 27 (10): 2141-9.
Disease progression and search for monogenic diabetes among children with new onset type 1 diabetes negative for ICA, GAD- and IA-2 Antibodies. , Pörksen S., BMC Endocr Disord. September 23, 2010; 10 16.
Investigations into the role of the Plasmodium falciparum SERCA (PfATP6) L263E mutation in artemisinin action and resistance. , Valderramos SG., Antimicrob Agents Chemother. September 1, 2010; 54 (9): 3842-52.
Aconitine blocks HERG and Kv1.5 potassium channels. , Li Y., J Ethnopharmacol. August 19, 2010; 131 (1): 187-95.
Alexa Fluor 546-ArIB[V11L;V16A] is a potent ligand for selectively labeling alpha 7 nicotinic acetylcholine receptors. , Hone AJ., J Neurochem. August 1, 2010; 114 (4): 994-1006.
Ginsenoside Rg3 activates human KCNQ1 K+ channel currents through interacting with the K318 and V319 residues: a role of KCNE1 subunit. , Choi SH., Eur J Pharmacol. July 10, 2010; 637 (1-3): 138-47.
[Inhibition of Jingzhaotoxin-V on Kv4.3 channel]. , Cai LJ., Sheng Li Xue Bao. June 25, 2010; 62 (3): 255-60.
Molecular determinants of Kv1.5 channel block by diphenyl phosphine oxide-1. , Du YM., J Mol Cell Cardiol. June 1, 2010; 48 (6): 1111-20.
Biochemical characterization of kappaM-RIIIJ, a Kv1.2 channel blocker: evaluation of cardioprotective effects of kappaM-conotoxins. , Chen P., J Biol Chem. May 14, 2010; 285 (20): 14882-14889.
Multiple mechanisms of hERG liability: K+ current inhibition, disruption of protein trafficking, and apoptosis induced by amoxapine. , Obers S., Naunyn Schmiedebergs Arch Pharmacol. May 1, 2010; 381 (5): 385-400.
A region of N-type Ca(2+) channel critical for blockade by the dihydropyridine amlodipine. , Miyashita Y., Eur J Pharmacol. April 25, 2010; 632 (1-3): 14-22.
Atypical alpha-conotoxin LtIA from Conus litteratus targets a novel microsite of the alpha3beta2 nicotinic receptor. , Luo S., J Biol Chem. April 16, 2010; 285 (16): 12355-66.
Block of the human ether-a- go-go-related gene ( hERG) K+ channel by the antidepressant desipramine. , Hong HK., Biochem Biophys Res Commun. April 9, 2010; 394 (3): 536-41.